Palladium-catalyzed ortho-acylation of 2-aryl pyridine derivatives using arylmethyl amines as new acyl sources.
نویسندگان
چکیده
A facile and efficient protocol for palladium-catalyzed ortho-acylation of 2-aryl pyridines was developed. Note that this acylation utilized arylmethyl amines as new, cheap and readily available acylation reagents and exhibited high regioselectivity for 2-aryl pyridines bearing a meta-substituent in the aryl ring moiety.
منابع مشابه
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ورودعنوان ژورنال:
- Chemical communications
دوره 49 61 شماره
صفحات -
تاریخ انتشار 2013